Four Cannabis Compounds Are Being Tested as Epilepsy Treatments

CBD has proven therapeutic benefit for Dravet and Lennox-Gastaut syndromes, while three other cannabinoids (CBDV, THCV, THCA) are in various stages of epilepsy research.

Ružić Zečević, Dejana et al.·Expert opinion on investigational drugs·2018·Moderate EvidenceReview
RTHC-01818ReviewModerate Evidence2018RETHINKTHC RESEARCH DATABASErethinkthc.com/research

Quick Facts

Study Type
Review
Evidence
Moderate Evidence
Sample
Not reported

What This Study Found

Preclinical studies confirmed anticonvulsant activity of CBD and CBDV across multiple epilepsy models. Clinical trials showed clear therapeutic benefit of CBD for treatment-resistant seizures in Dravet syndrome and drop seizures in Lennox-Gastaut syndrome, with good safety profiles.

Key Numbers

Four cannabinoids investigated: CBD, CBDV, THCV, and THCA. CBD showed benefit specifically in Dravet syndrome and Lennox-Gastaut syndrome (LGS). Clinical trials for CBDV results were still pending at publication.

How They Did This

Review of preclinical and clinical studies on investigational cannabinoids for epilepsy, searched across MEDLINE, SCOPUS, EBSCO, Google Scholar, and SCINDEX databases.

Why This Research Matters

About one-third of epilepsy patients are drug-resistant. CBD has become the first cannabis-derived compound approved for epilepsy, and several other cannabinoids in the research pipeline could expand treatment options.

The Bigger Picture

The success of CBD for epilepsy has opened the door for investigating other cannabinoids. Each compound has different mechanisms of action, which could mean different cannabinoids work for different types of seizures.

What This Study Doesn't Tell Us

Clinical evidence was strongest for CBD; other cannabinoids still lacked human trial data. The full therapeutic potential across epilepsy types remains unknown.

Questions This Raises

  • ?Will CBDV clinical trials show the same promise as preclinical data suggested?
  • ?Could combinations of cannabinoids be more effective than single compounds?
  • ?What mechanisms explain CBD's anticonvulsant effects?

Trust & Context

Key Stat:
One-third of epilepsy patients are drug-resistant; CBD showed clear benefit for the most severe pediatric forms.
Evidence Grade:
Moderate - review covers both established (CBD) and preliminary (other cannabinoids) evidence with appropriate distinction between the two.
Study Age:
Published in 2018. CBD (Epidiolex) has since been FDA-approved for these indications.
Original Title:
Investigational cannabinoids in seizure disorders, what have we learned thus far?
Published In:
Expert opinion on investigational drugs, 27(6), 535-541 (2018)
Database ID:
RTHC-01818

Evidence Hierarchy

Meta-Analysis / Systematic Review
Randomized Controlled Trial
Cohort / Case-Control
Cross-Sectional / ObservationalSnapshot without intervening
This study
Case Report / Animal Study

Summarizes existing research on a topic.

What do these levels mean? →

Frequently Asked Questions

Does CBD help with seizures?

Clinical trials showed clear therapeutic benefit of CBD for treatment-resistant seizures in Dravet syndrome and Lennox-Gastaut syndrome. It has since been FDA-approved for these conditions as Epidiolex.

Are there other cannabis compounds that might treat epilepsy?

Three other cannabinoids are being investigated: CBDV (cannabidivarin), THCV, and THCA. Preclinical data is promising, but human trial data was still limited at the time of this review.

Read More on RethinkTHC

Cite This Study

RTHC-01818·https://rethinkthc.com/research/RTHC-01818

APA

Ružić Zečević, Dejana; Folić, Marko; Tantoush, Ziyad; Radovanović, Milan; Babić, Goran; Janković, Slobodan M. (2018). Investigational cannabinoids in seizure disorders, what have we learned thus far?. Expert opinion on investigational drugs, 27(6), 535-541. https://doi.org/10.1080/13543784.2018.1482275

MLA

Ružić Zečević, Dejana, et al. "Investigational cannabinoids in seizure disorders, what have we learned thus far?." Expert opinion on investigational drugs, 2018. https://doi.org/10.1080/13543784.2018.1482275

RethinkTHC

RethinkTHC Research Database. "Investigational cannabinoids in seizure disorders, what have..." RTHC-01818. Retrieved from https://rethinkthc.com/research/ruzic-2018-investigational-cannabinoids-in-seizure

Access the Original Study

Study data sourced from PubMed, a service of the U.S. National Library of Medicine, National Institutes of Health.

This study breakdown was produced by the RethinkTHC research team. We analyze and report published research findings without making health recommendations. All interpretations are based solely on the published abstract and study data.