Cannabis extracts produced different pain relief than pure THC-CBD blends at the same ratio

A whole-plant cannabis extract and a pure 1:1 THC:CBD mixture produced distinct pain-relief profiles and engaged different endocannabinoid targets in a rat model of diabetic neuropathy, despite having the same THC:CBD ratio.

Benredjem, Besma et al.·Frontiers in pharmacology·2023·Preliminary EvidenceAnimal StudyAnimal Study
RTHC-04410Animal StudyPreliminary Evidence2023RETHINKTHC RESEARCH DATABASErethinkthc.com/research

Quick Facts

Study Type
Animal Study
Evidence
Preliminary Evidence
Sample
Not reported

What This Study Found

When injected into the spinal fluid of rats with diabetic neuropathy, a type II cannabis extract and a 1:1 THC:CBD mix produced different antinociceptive responses despite equivalent THC content. The two preparations also engaged CB1, CB2 receptors, and TRPV1 channels differently.

Key Numbers

Four conditions tested: pure THC, pure CBD, 1:1 THC:CBD mix, balanced extract; three receptor systems evaluated (CB1, CB2, TRPV1)

How They Did This

Animal study using a rat model of diabetic neuropathy with intrathecal injection of pure THC, pure CBD, a 1:1 THC:CBD mix, and a balanced chemotype II cannabis extract. Receptor involvement assessed using CB1, CB2, and TRPV1 antagonists.

Why This Research Matters

Current medical cannabis prescribing relies heavily on THC:CBD ratios to predict effects. This study suggests that the full composition of an extract matters, not just its major cannabinoid ratio.

The Bigger Picture

The finding that same-ratio preparations produce different effects supports the entourage effect concept and challenges the practice of categorizing medical cannabis products primarily by THC:CBD ratio.

What This Study Doesn't Tell Us

Animal model with intrathecal (spinal) delivery, which does not reflect typical human routes of administration. Diabetic neuropathy model may not generalize to other pain types. Single extract tested.

Questions This Raises

  • ?Which minor cannabinoids or terpenes in the whole-plant extract account for the different receptor engagement?
  • ?Would these differences hold with oral or inhaled administration?

Trust & Context

Key Stat:
Same THC:CBD ratio, different pain relief profiles and receptor targets
Evidence Grade:
Animal study with controlled conditions and receptor-level analysis, but spinal delivery route and single extract tested limit clinical translation.
Study Age:
Published 2023
Original Title:
A type II cannabis extract and a 1:1 blend of Δ(9)-tetrahydrocannabinol and cannabidiol display distinct antinociceptive profiles and engage different endocannabinoid targets when administered into the subarachnoid space.
Published In:
Frontiers in pharmacology, 14, 1235255 (2023)
Database ID:
RTHC-04410

Evidence Hierarchy

Meta-Analysis / Systematic Review
Randomized Controlled Trial
Cohort / Case-Control
Cross-Sectional / Observational
Case Report / Animal StudyOne case or non-human subjects
This study

Tests effects in animals (usually mice or rats), not humans.

What do these levels mean? →

Frequently Asked Questions

Does the THC:CBD ratio predict how a cannabis product will work?

This animal study suggests not entirely. A whole cannabis extract and a pure 1:1 THC:CBD blend produced different pain relief responses and activated different receptor systems despite having the same ratio.

What is the entourage effect?

The idea that compounds in cannabis work together, so whole-plant extracts may produce different effects than isolated cannabinoids. This study provides evidence supporting that concept.

Read More on RethinkTHC

Cite This Study

RTHC-04410·https://rethinkthc.com/research/RTHC-04410

APA

Benredjem, Besma; Pineyro, Graciela. (2023). A type II cannabis extract and a 1:1 blend of Δ(9)-tetrahydrocannabinol and cannabidiol display distinct antinociceptive profiles and engage different endocannabinoid targets when administered into the subarachnoid space.. Frontiers in pharmacology, 14, 1235255. https://doi.org/10.3389/fphar.2023.1235255

MLA

Benredjem, Besma, et al. "A type II cannabis extract and a 1:1 blend of Δ(9)-tetrahydrocannabinol and cannabidiol display distinct antinociceptive profiles and engage different endocannabinoid targets when administered into the subarachnoid space.." Frontiers in pharmacology, 2023. https://doi.org/10.3389/fphar.2023.1235255

RethinkTHC

RethinkTHC Research Database. "A type II cannabis extract and a 1:1 blend of Δ(9)-tetrahydr..." RTHC-04410. Retrieved from https://rethinkthc.com/research/benredjem-2023-a-type-ii-cannabis

Access the Original Study

Study data sourced from PubMed, a service of the U.S. National Library of Medicine, National Institutes of Health.

This study breakdown was produced by the RethinkTHC research team. We analyze and report published research findings without making health recommendations. All interpretations are based solely on the published abstract and study data.