Repeated exposure to a synthetic cannabinoid caused lasting cognitive and brain changes in mice

Seven days of JWH-018 exposure in mice produced psychotic-like symptoms and lasting impairments in memory, social behavior, and brain plasticity that persisted for at least 15 days after the drug was stopped.

Bilel, Sabrine et al.·British journal of pharmacology·2023·Preliminary EvidenceAnimal StudyAnimal Study
RTHC-04417Animal StudyPreliminary Evidence2023RETHINKTHC RESEARCH DATABASErethinkthc.com/research

Quick Facts

Study Type
Animal Study
Evidence
Preliminary Evidence
Sample
Not reported

What This Study Found

Repeated JWH-018 treatment (6 mg/kg daily for 7 days) induced psychomotor agitation, reduced social dominance and recognition memory, impaired prepulse inhibition, disrupted hippocampal long-term potentiation, decreased BDNF expression, and altered endocannabinoid system components in the striatum and hippocampus, all persisting 15+ days after last exposure.

Key Numbers

6 mg/kg JWH-018 daily for 7 days; 15-16 day washout; reduced hippocampal CB1 receptor density; altered AEA and 2-AG levels; decreased BDNF, PSD95, and NMDA receptor subunit expression

How They Did This

Male CD-1 mice received daily injections of vehicle, JWH-018 (6 mg/kg), CB1 antagonist NESS-0327 (1 mg/kg), or co-administration for 7 days. After 15-16 days washout, behavioral, neurochemical, electrophysiological, and molecular assessments were performed.

Why This Research Matters

Synthetic cannabinoids are far more potent than plant cannabis and are associated with severe psychiatric outcomes in humans. This study provides mechanistic evidence for how repeated exposure produces lasting brain changes.

The Bigger Picture

The persistence of cognitive and neuroplasticity deficits well after drug cessation raises concerns about lasting brain damage from synthetic cannabinoid use, which is particularly relevant given the prevalence of these substances in unregulated markets.

What This Study Doesn't Tell Us

Used a single high dose in male mice only. JWH-018 is one of many synthetic cannabinoids with varying potency. Route of administration (injection) differs from typical human use (smoking). No female mice included.

Questions This Raises

  • ?Are these neuroplasticity changes reversible with longer washout periods?
  • ?Do lower doses or intermittent exposure produce similar lasting effects?

Trust & Context

Key Stat:
Cognitive and brain changes persisted 15+ days after stopping the drug
Evidence Grade:
Well-designed animal study with multiple outcome measures and CB1 antagonist control, but single dose level in male mice only limits generalizability.
Study Age:
Published 2023
Original Title:
Cognitive dysfunction and impaired neuroplasticity following repeated exposure to the synthetic cannabinoid JWH-018 in male mice.
Published In:
British journal of pharmacology, 180(21), 2777-2801 (2023)
Database ID:
RTHC-04417

Evidence Hierarchy

Meta-Analysis / Systematic Review
Randomized Controlled Trial
Cohort / Case-Control
Cross-Sectional / Observational
Case Report / Animal StudyOne case or non-human subjects
This study

Tests effects in animals (usually mice or rats), not humans.

What do these levels mean? →

Frequently Asked Questions

How do synthetic cannabinoids affect the brain differently than plant cannabis?

This study found that repeated JWH-018 (a synthetic cannabinoid) exposure caused lasting changes to memory, social behavior, brain plasticity, and the endocannabinoid system itself. These effects persisted at least 15 days after the drug was stopped.

Were the cognitive effects reversible?

After 15-16 days without the drug, mice still showed impaired memory, reduced social dominance, disrupted brain plasticity, and altered endocannabinoid signaling. Whether longer recovery periods would allow reversal was not tested.

Read More on RethinkTHC

Cite This Study

RTHC-04417·https://rethinkthc.com/research/RTHC-04417

APA

Bilel, Sabrine; Zamberletti, Erica; Caffino, Lucia; Tirri, Micaela; Mottarlini, Francesca; Arfè, Raffaella; Barbieri, Mario; Beggiato, Sarah; Boccuto, Federica; Bernardi, Tatiana; Casati, Sara; Brini, Anna T; Parolaro, Daniela; Rubino, Tiziana; Ferraro, Luca; Fumagalli, Fabio; Marti, Matteo. (2023). Cognitive dysfunction and impaired neuroplasticity following repeated exposure to the synthetic cannabinoid JWH-018 in male mice.. British journal of pharmacology, 180(21), 2777-2801. https://doi.org/10.1111/bph.16164

MLA

Bilel, Sabrine, et al. "Cognitive dysfunction and impaired neuroplasticity following repeated exposure to the synthetic cannabinoid JWH-018 in male mice.." British journal of pharmacology, 2023. https://doi.org/10.1111/bph.16164

RethinkTHC

RethinkTHC Research Database. "Cognitive dysfunction and impaired neuroplasticity following..." RTHC-04417. Retrieved from https://rethinkthc.com/research/bilel-2023-cognitive-dysfunction-and-impaired

Access the Original Study

Study data sourced from PubMed, a service of the U.S. National Library of Medicine, National Institutes of Health.

This study breakdown was produced by the RethinkTHC research team. We analyze and report published research findings without making health recommendations. All interpretations are based solely on the published abstract and study data.